Philpott, Carl
Carl Philpott
VIAF ID: 308757649 (Personal)
Permalink: http://viaf.org/viaf/308757649
Preferred Forms
- 100 0 _ ‡a Carl Philpott
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- 100 1 _ ‡a Philpott, Carl
- 100 1 _ ‡a Philpott, Carl
4xx's: Alternate Name Forms (2)
Works
Title | Sources |
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[1,2,4]triazolo[4,3-a]phthalazines: inhibitors of diverse bromodomains | |
3,5-dimethylisoxazoles act as acetyl-lysine-mimetic bromodomain ligands | |
Bromodomain-peptide displacement assays for interactome mapping and inhibitor discovery | |
Bullet points in ENT, 2014: | |
The design and synthesis of 5- and 6-isoxazolylbenzimidazoles as selective inhibitors of the BET bromodomains | |
Generation of a Selective Small Molecule Inhibitor of the CBP/p300 Bromodomain for Leukemia Therapy | |
Identification of a Chemical Probe for Bromo and Extra C-Terminal Bromodomain Inhibition through Optimization of a Fragment-Derived Hit | |
PFI-1, a highly selective protein interaction inhibitor, targeting BET Bromodomains | |
RVX-208, an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain | |
A series of potent CREBBP bromodomain ligands reveals an induced-fit pocket stabilized by a cation-π interaction |