Thomas Durek researcher
Durek, Thomas
VIAF ID: 2687153954868905680004 (Personal)
Permalink: http://viaf.org/viaf/2687153954868905680004
Preferred Forms
- 100 1 _ ‡a Durek, Thomas
- 100 0 _ ‡a Thomas Durek ‡c researcher
4xx's: Alternate Name Forms (3)
5xx's: Related Names (2)
Works
Title | Sources |
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Analgesic Effects of GpTx-1, PF-04856264 and CNV1014802 in a Mouse Model of NaV1.7-Mediated Pain. | |
Approaches to the stabilization of bioactive epitopes by grafting and peptide cyclization. | |
A bifunctional asparaginyl endopeptidase efficiently catalyzes both cleavage and cyclization of cyclic trypsin inhibitors | |
A Centipede Toxin Family Defines an Ancient Class of CSαβ Defensins | |
Characterisation of Na(v) types endogenously expressed in human SH-SY5Y neuroblastoma cells | |
Characterization of Synthetic Tf2 as a NaV1.3 Selective Pharmacological Probe | |
Chemical synthesis, 3D structure, and ASIC binding site of the toxin mambalgin-2 | |
Chemical synthesis and folding of APETx2, a potent and selective inhibitor of acid sensing ion channel 3. | |
Combining Sense and Nonsense Codon Reassignment for Site-Selective Protein Modification with Unnatural Amino Acids. | |
Constrained Cyclic Peptides as Immunomodulatory Inhibitors of the CD2:CD58 Protein-Protein Interaction | |
Convergent chemical synthesis and high-resolution x-ray structure of human lysozyme | |
Cyclic alpha-conotoxin peptidomimetic chimeras as potent GLP-1R agonists | |
Development of Novel Melanocortin Receptor Agonists Based on the Cyclic Peptide Framework of Sunflower Trypsin Inhibitor-1. | |
The E15R Point Mutation in Scorpion Toxin Cn2 Uncouples Its Depressant and Excitatory Activities on Human NaV1.6. | |
Europium-Labeled Synthetic C3a Protein as a Novel Fluorescent Probe for Human Complement C3a Receptor | |
Fmoc-based synthesis of disulfide-rich cyclic peptides. | |
Highly Potent and Selective Plasmin Inhibitors Based on the Sunflower Trypsin Inhibitor-1 Scaffold Attenuate Fibrinolysis in Plasma | |
Intein-mediated synthesis of geranylgeranylated Rab7 protein in vitro | |
Interaction of Synthetic Human SLURP-1 with the Nicotinic Acetylcholine Receptors. | |
Isolation and structural and pharmacological characterization of α-elapitoxin-Dpp2d, an amidated three finger toxin from black mamba venom | |
Isolation of two insecticidal toxins from venom of the Australian theraphosid spider Coremiocnemis tropix. | |
Isolation, synthesis and characterization of ω-TRTX-Cc1a, a novel tarantula venom peptide that selectively targets L-type Cav channels | |
Mapping of voltage sensor positions in resting and inactivated mammalian sodium channels by LRET. | |
Modulation of human Nav1.7 channel gating by synthetic α-scorpion toxin OD1 and its analogs | |
Molecular basis for the production of cyclic peptides by plant asparaginyl endopeptidases. | |
Neurotoxic peptides from the venom of the giant Australian stinging tree | |
Nicotiana alata Defensin Chimeras Reveal Differences in the Mechanism of Fungal and Tumor Cell Killing and an Enhanced Antifungal Variant | |
NMR Structure of μ-Conotoxin GIIIC: Leucine 18 Induces Local Repacking of the N-Terminus Resulting in Reduced Na Channel Potency | |
Papain-like cysteine proteases prepare plant cyclic peptide precursors for cyclization | |
Phage display-based discovery of cyclic peptides against the broad spectrum bacterial anti-virulence target CsrA | |
Potent complement C3a receptor agonists derived from oxazole amino acids: Structure-activity relationships. | |
Preformed selenoesters enable rapid native chemical ligation at intractable sites | |
Protein semi-synthesis: new proteins for functional and structural studies. | |
Site-Specific Sequential Protein Labeling Catalyzed by a Single Recombinant Ligase | |
Structure of doubly prenylated Ypt1:GDI complex and the mechanism of GDI-mediated Rab recycling | |
Structure of Rab GDP-dissociation inhibitor in complex with prenylated YPT1 GTPase | |
A suite of kinetically superior AEP ligases can cyclise an intrinsically disordered protein | |
Synthesis of fluorescently labeled mono- and diprenylated Rab7 GTPase | |
Synthesis of Functionalized Rab GTPases by a Combination of Solution- or Solid-Phase Lipopeptide Synthesis with Expressed Protein Ligation | |
Synthesis of photoactive analogues of a cystine knot trypsin inhibitor protein | |
The tarantula toxin β/δ-TRTX-Pre1a highlights the importance of the S1-S2 voltage-sensor region for sodium channel subtype selectivity. | |
Targeted Delivery of Cyclotides via Conjugation to a Nanobody | |
Therapeutic conotoxins: a US patent literature survey | |
Total chemical synthesis, folding, and assay of a small protein on a water-compatible solid support | |
Two for the Price of One: Heterobivalent Ligand Design Targeting Two Binding Sites on Voltage-Gated Sodium Channels Slows Ligand Dissociation and Enhances Potency |