Boumendjel, Ahcène 1964-..
Ahcène Boumendjel researcher
Boumendjel, Ahcène
VIAF ID: 86277907 (Personal)
Permalink: http://viaf.org/viaf/86277907
Preferred Forms
- 100 0 _ ‡a Ahcène Boumendjel ‡c researcher
- 100 1 _ ‡a BOUMENDJEL, AHCENE.
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- 100 1 _ ‡a Boumendjel, Ahcène
- 100 1 _ ‡a Boumendjel, Ahcène, ‡d 1964-....
- 100 1 _ ‡a Boumendjel, Ahcène ‡d 1964-..
4xx's: Alternate Name Forms (1)
Works
Title | Sources |
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2-Arylidenedihydroindole-3-ones: design, synthesis, and biological activity on bladder carcinoma cell lines. | |
2-Indolylmethylenebenzofuranones as first effective inhibitors of ABCC2. | |
3-Aryl-4-methyl-2-quinolones targeting multiresistant Staphylococcus aureus bacteria. | |
ABC transporters and multidrug resistance, c2009: | |
ABCG2: recent discovery of potent and highly selective inhibitors | |
Analogues de flavonoïdes inhibiteurs de la glycoprotéine P, modulateurs potentiels de la chimiorésistance | |
Antiviral and immunomodulatory activity of alkaloids against infection by the arthritogenic alphavirus O'nyong-nyong. | |
Application de la synthèse de Weinreb des aldéhydes à la synthèse totale d'alcaloïdes indoliques | |
Are Human Tyrosinase and Related Proteins Suitable Targets for Melanoma Therapy? | |
Arylthiosemicarbazones as antileishmanial agents | |
Breast cancer resistance protein (BCRP/ABCG2): new inhibitors and QSAR studies by a 3D linear solvation energy approach. | |
Caractérisation biochimique de YphC, une protéine de Bacillus subtilis à deux domaines GTPases impliquée dans la biogenèse du ribosome | |
Cellular and molecular mechanisms activating the cell death processes by chalcones: Critical structural effects | |
Chalcone JAI-51 improves efficacy of synchrotron microbeam radiation therapy of brain tumors. | |
Chalcones derivatives acting as cell cycle blockers: potential anti cancer drugs? | |
Conception, synthèse et évalutation de prodrogues à espaceurs clivables : application à la chimiothérapie vectorisée du mélanome | |
Contribution to the study of the natural origin of tramadol and phytochemical study of two alpine plants. | |
Design, synthèse et caractérisation d'inhibiteurs d'hélicase Pif1 et BLM | |
Design, synthesis and biological activity of peptidic vectors for the diagnostic and/or therapy of tumours. | |
Design, synthesis and biological evaluations of quinoxalines and analogues as Pim-1 kinase inhibitors. | |
Design, synthesis and evaluation of prodrugs with cleavable linkers : application to targeted chemotherapy of metastatic melanoma. | |
Design, Synthesis and Evaluation of the antimitotic effect of 2-phenyl-4-quinolones. | |
Dicer-mediated upregulation of BCRP confers tamoxifen resistance in human breast cancer cells | |
The effect of flavonoid derivatives on doxorubicin transport and metabolism. | |
Efficient approach to thapsigargins (guaianolides) and synthesis of red azulenes via a common intermediate bicyclo[5.3.0]decane. | |
Flavonoids as RTK inhibitors and potential anticancer agents | |
General Articles Aurones: A Subclass of Flavones with Promising Biological Potential | |
Les hydrocabures aromatiques polycycliques : un problème de santé publique | |
Identification, physico-chemical and pharmacological characterizations of a new melanogenesis inhibitor, isolated from animal venoms : argiotoxin-636 example. | |
Inhibiteurs du transporteur BCRP/ABCG2 impliqué dans la chimiorésistance : conception, synthèse et évaluation biologique | |
Investigation of a new 1,3-diarylpropenone as a potential antimitotic agent targeting bladder carcinoma. | |
IPP51, a chalcone acting as a microtubule inhibitor with in vivo antitumor activity against bladder carcinoma | |
Lien entre le cannabis médicinal et l'axe de signalisation autotaxine acide lysophosphatidique : développement d'inhibiteurs inspirés des cannabinoïdes | |
MBL-II-141, a chromone derivative, enhances irinotecan (CPT-11) anticancer efficiency in ABCG2-positive xenografts | |
Modulation of paclitaxel transport by flavonoid derivatives in human breast cancer cells. Is there a correlation between binding affinity to NBD of P-gp and modulation of transport? | |
Multicomponent synthesis and pharmacological evaluation of multi-targeted directed Ligand via Ugi and Hantzsch reactions as a solution for Alzheimer's disease.. | |
Nauclea latifolia: biological activity and alkaloid phytochemistry of a West African tree | |
A novel chalcone derivative which acts as a microtubule depolymerising agent and an inhibitor of P-gp and BCRP in in-vitro and in-vivo glioblastoma models | |
A Novel Platinum-Maurocalcine Conjugate Induces Apoptosis of Human Glioblastoma Cells by Acting through the ROS-ERK/AKT-p53 Pathway. | |
Occurrences, biosynthesis and properties of aurones as high-end evolutionary products. | |
Optimization of the chromone scaffold through QSAR and docking studies: Identification of potent inhibitors of ABCG2 | |
Ovarian cancer cells cisplatin sensitization agents selected by mass cytometry target ABCC2 inhibition | |
Phytochemical analyses and anti-inflammatory activities of medicinal plants from the Auvergne region. | |
Phytochemical and Biological Investigation of Helianthemum nummularium, a High-Altitude Growing Alpine Plant Overrepresented in Ungulates Diets | |
Piperidinyl-embeded chalcones possessing anti PI3Kδ inhibitory properties exhibit anti-atopic properties in preclinical models | |
Quantitative evaluation of the combination between cytotoxic drug and efflux transporter inhibitors based on a tumour growth inhibition model. | |
Recent advances in the discovery of flavonoids and analogs with high-affinity binding to P-glycoprotein responsible for cancer cell multidrug resistance. | |
Recherche et étude de molécules à activité antityrosinase et leur utilisation comme agents dépigmentants en dermocosmétique | |
A retro-biosynthetic approach to the prediction of biosynthetic pathways from position-specific isotope analysis as shown for tramadol | |
Search and investigation of tyrosinase inhibitor and their potent use in dermocosmetics. | |
Structure-activity relationships in the development of allosteric hepatitis C virus RNA-dependent RNA polymerase inhibitors: ten years of research | |
Structure-activity relationships of chromone derivatives toward the mechanism of interaction with and inhibition of breast cancer resistance protein ABCG2. | |
Study and Optimisation of Immunogenic Compounds and Multidrug Resistance Modulators by Molecular Modeling Technics. | |
Substituted chromones as highly potent nontoxic inhibitors, specific for the breast cancer resistance protein | |
Synthèse de 5- et 6-azaindoles, de stéroïdes et de composés divalents adénine-stéroïdes : évaluation de l'effet modulateur vis-à-vis de la glycoprotéine P | |
Synthèse de nouveaux détergents extractants et stabilisants des protéines membranaireset synthèse de dérivés d'aurones comme inhibiteurs d'ABCC2 | |
Synthèse d'inhibiteurs de l'interaction entre la protéine à domaine PDZ, PSD-95 et le récepteur de la sérotoninte 5-HT2A pour le traitement des douleurs neuropathiques | |
Synthèse et évaluation biologique de dérivés hétérocyliques comme agents anti-cancéreux | |
Synthèse et évaluation d'aurones sur des modèles de fibres de tau | |
Synthèse multicomposants et évaluation pharmacologique de molécules multicibles par des réactions d'Ugi et de Hantzsch comme solution pour la maladie d'Alzheimer | |
Synthèses de bis(hétéroaryl)alcanes et de pyrrolyl méthanamines chirales. | |
Synthesis of alkaloids of the Lycorine family through tandem ring closing metathesis. | |
Synthesis of biomoleculesactingas inhibitors ofRNA-dependent RNA polymerase ofhepatitis Cvirus and development of novel generation of surfactants acting as membrane proteins stabilizers. | |
A synthetic chalcone as a potent inducer of glutathione biosynthesis | |
Targeting the Achilles heel of multidrug-resistant cancer by exploiting the fitness cost of resistance | |
Techniques de Modélisation Moléculaire appliquées à l’Etude et à l’Optimisation de Molécules Immunogènes et de Modulateurs de la Chimiorésistance | |
A template model for studying anticancer drug efflux transporter inhibitors in vitro | |
Therapeutic iontophoresis for scleroderma-related cutaneous ulcerations : screening, proof-of-concept study in a mouse scleroderma model. | |
Toward a therapy for two rare vascular diseases : screenings of medical chemo-libraries for Rendu-Osler Disease and Pulmonary Arterial Hypertension. | |
Traditional uses, phytochemistry and pharmacological properties of African Nauclea species: A review | |
Transmission d’un bilan de secours et mise en place de protocoles de soins d’urgence pour le pharmacien d’officine | |
Le transporteur ABCG2 de multiples drogues : rôle d'une séquence spécifique et recherche d'inhibiteurs sélectifs | |
Two in one: bifonctional derivatives of trolox acting as antimalarial and antioxidant agents | |
Validation d'une méthode de déréplication de substances naturelles marines | |
Validation of a marine natural products dereplication strategy. | |
Vers une thérapie pour deux maladies vasculaires rares : criblage de chimiothèques de médicaments pour les maladies Rendu-Osler et Hypertension Artérielle Pulmonaire |